Thanzi, Kukonzekera
"Thiotriazoline": malangizo ntchito
Kodi inu kulemba mankhwala "Thiotriazoline"? kugwiritsa ntchito bukuli mankhwala adzakhala anafotokoza m'nkhani pano. Komanso, ife tinena za mtundu umene mankhwala akulowa zogulitsa anati, umene ali zizindikiro, mavuto ndi contraindications.
The zikuchokera kwa ma CD mankhwala ndi mawonekedwe kumasulidwa
Kodi maonekedwe kumasulidwa medicament "Thiotriazoline"? Malangizo imatiuza kuti amagwiritsa ntchito zosiyanasiyana. Wotchuka kwambiri ndi:
- A njira anafuna mu mnofu ndi mtsempha jekeseni. 1 ml ya wothandizila lili 0,025 ga Thiotriazoline. Komanso medicament ndi mbali optional mu mawonekedwe a madzi a jekeseni. Mankhwala akupezeka 4 ml ya ampoules (anaikidwa katoni).
- "Thiotriazoline" m'maso. Mwa kugwiritsa ntchito kalozera zikutanthauza imafotokoza kuti 5 ml ya lili 50 mg wa mankhwala Thiotriazoline, komanso zinthu zina. Mankhwala chogulitsidwa mabotolo pulasitiki, droppers, anaika mukatoni.
- "Thiotriazoline" mankhwala. Malangizo kwa mawonekedwe ya mankhwala imafotokoza kuti mu woyera mapiritsi zozungulira ndi lathyathyathya pamwamba munali 100 mg morfoliniymetiltriazoliltioatsetata, kapena otchedwa Thiotriazoline. Monga zigawo zina za medicament zimene mbatata wowuma, microcrystalline mapadi, otsika maselo kulemera povidone, calcium stearate ndi sucrose. Monga ulamuliro, mu phukusi makatoni lili mapiritsi 50.
pharmacodynamics
ndi mankhwala monga "Thiotriazoline" n'chiyani? Malangizo Ntchito limanena kuti mankhwala antioxidant. imachita yapamwamba chifukwa antioxidant, antiischemic, immunomodulatory ndi Kakhungu ofunika katundu.
Ankaona mankhwala kumathandiza chiwonongeko cha hepatocytes, zimathandiza kuchira awo, kuchepetsa mlingo wa mafuta kusalola, chifukwa mu normalization zomanga thupi, zimam'patsa zamadzimadzi ndi pigment kuwombola, ndipo kumachepetsa mosavuta kufala kwa necrosis tsentrolobulyarnyh thupi monga chiwindi. Komanso, yogwira mankhwala bwino payekha kaphatikizidwe ya ndulu, normalizes kapangidwe kake (mankhwala).
The katundu wa mankhwala
Kodi katundu wa mankhwala "Thiotriazoline"? Malangizo ntchito mankhwala chofunika kuwerenga. Ndipotu yekha kwa inu mukhoza kuphunzira zimene mankhwala ankaona Sachita chopinga zako zobwera chifukwa cha okosijeni mu za Krebs adzizungulira, kusunga okhudza maselo ambiri ATP thumba, komanso timapitiriza kutsegula (compensatory) anaerobic glycolysis.
Amanenanso kuti kutenga mankhwala yogwira chinthu akuyamba yambitsa dongosolo antioxidant, mafuta ziletsa njira zobwera chifukwa cha okosijeni m'madera ischemic za thupi. Komanso, mankhwala bwino katundu (rheology) ya magazi chifukwa kutsegula a dongosolo fibrinolytic.
The antioxidant katundu wa mankhwala anaonetsa chakuti kapangidwe ka molekyulu ndi tiotrazolina ayoni sulfure, yodziwika ndi makutidwe ndi okosijeni ndi kuchepetsa zinthu, komanso ukachenjede asafe, amene chimango ndi yambiri ya ayoni wa hydrogen.
Tiyenera kuona kuti yogwira chigawo mankhwala akhoza kutani ndi ankafuna kusintha zinthu mopitirira zamadzimadzi ndi mitundu zotakasika mpweya. Ichi ndi chifukwa ndi kutchulidwa katundu kuchepetsa gulu thiol. Komanso, medicament kumathandiza mapangidwe mitundu zotakasika mpweya, monga antiradical reactivating michere monga catalase, glutathione peroxidase ndi superoxide dismutase.
Pharmacokinetics
Kaya mankhwala odzipereka "Thiotriazoline"? Malangizo limanena kuti nthawi poluabsorbtsii mankhwala mphindi 30 ndi bioavailability - 65,5%.
Zolemba malire ndende magazi kudzera Zimapezeka maola 1.4 pambuyo utsogoleli. Kulankhulana ndi mapuloteni si upambana 10%.
Lalikulu zedi, mankhwala amasonkhana mu zimakhala a chiwindi, mtima, m'matumbo, ndulu ndi impso, ndi zazing'ono - mu intestine ang'ono ndi mapapo. Thiotriazoline excreted makamaka ndi impsozo.
umboni
Ngati pali zolakwika awerenge mankhwala, jakisoni ndi diso akutsikira "Thiotriazoline"? kugwiritsa ntchito mitundu imeneyi ya malangizo zikusonyeza zizindikiro zotsatirazi:
- matenda enaake;
- poizoni chiwindi kuwonongeka, mowa, tizilombo, ndi mankhwala (mwachitsanzo, atalandira mankhwala mavairasi oyambitsa mankhwala, odana ndi TB ndi odana ndi chotupa wothandizira, kulera m'kamwa ndi antidepressants tricyclic);
- aakulu tizilombo matenda a chiwindi;
- mowa chiwindi aakulu zolimbitsa ntchito kochepa;
- mafuta m'chiwindi alibe.
Zikuonetsa ntchito madontho:
- matenda corneal;
- zilonda zamoto kapena diso kuvulala;
- tizilombo conjunctivitis.
Chifukwa kugwiritsira ntchito ophthalmic mankhwala "Thiotriazoline"? Malangizo (madontho lingathe kukopedwa pa ogulitsa mankhawala aliyense) imatiuza kuti mankhwala kawirikawiri analamula kuti kupewa msozi, eyestrain, ndi matenda ena yotupa ziwalo zithunzi.
Miyala mlingo
Kodi ndimagwiritsa ntchito "Thiotriazoline" piritsi? Buku lili ndi mfundo zimene mankhwala ayenera kumwedwa mkati yekha. Monga ulamuliro, thiotriazolin anaika piritsi 1 kapena 2 kanayi pa tsiku kwa masiku 25-30.
Kutalika kwa mankhwala ndi wothandizila ichi tiyenera kuyesetsa ndi dokotala pa maziko munthu (malingana Inde ndiponso azikhala matenda wogwila).
The njira mankhwala "Thiotriazoline": malangizo ntchito
Majekeseni "Thiotriazoline" kuchita intramuscularly kapena kudzera m'mitsempha. mlingo awo anatsimikiza ndi dokotala (malingana ndi matenda). M'mnyewa wamtima infarction ndi chiwindi mankhwala pang'onopang'ono jekeseni kudzera m'mitsempha mu 2 ml 2-3 pa tsiku. Mu matenda enaake medicament chikuyendetsedwera intramuscularly (2 ml 2-3 nthawi tsiku). The njira ya mankhwala masiku 60.
M'maso "Thiotriazoline": malangizo ntchito
M'maso "Thiotriazoline" anaika mu sac conjunctival. Kawirikawiri, mlingo akuluakulu 2 madontho nthawi mpaka 4 tsiku. Pankhani ana, kuchuluka kwa mankhwala anatsimikiza yekha ndi dokotala wa ana. Kutalika kwa mankhwala ndi madontho diso ndipo iyenera kukhazikitsidwa ndi dokotala nawo.
Monga ulamuliro, nthawi ya mankhwala ndi chida ichi palibe kuposa 2 masabata. Koma ngati palibe kusintha zimawonedwa, ndithudi angathe mwezi wathunthu.
Ngati zotupa yaikulu ziwalo zithunzi ndi lalikulu, ndiyeno dropwise Kuwonjezera jakisoni ocular kutumikiridwa (kukonzekera taphunzira).
Pakuti kupewa kuyanika wa nembanemba diso (pamene ntchito pa kompyuta), muyenera kugwiritsa ntchito mankhwala 2 madontho masana ndi imeneyi ya maola 2.
zotsatira zoyipazi
Kodi mavuto a mankhwala zingachititse "Thiotriazoline" (akatemera)? Malangizo kwa njira imeneyi zikusonyeza kuti mankhwala ndi bwino analekerera ndi ulemu. Komabe, pogwiritsa ntchito mankhwala ankaona akhoza zimachitika zochita zoipa.
- Chapakati mantha dongosolo: chizungulire, kufooka, kulira m'khutu.
- M'mimba thirakiti: pakamwa youma, nseru, bloating.
- Ziwiya ndi mtima, kuthamanga magazi, tachycardia, arrhythmia, kupweteka mtima.
- Kupuma dongosolo: mphumu ndi kupuma movutikira.
- Ziwengo: malungo, zochita hypersensitivity, angioedema.
- zochita Local: redness ndi kumva kulasalasa kutengeka pa malo jekeseni.
- zochita Dermatological: ankatenthetsa khungu, kuyabwa, ming'oma.
Koma madontho diso, pa gawo lawo mavuto amene anaona.
Mwanjira mankhwala
Malinga ndi akatswiri, mankhwala "Thiotriazoline" angagwiritsidwe ntchito molumikizana ndi mankhwala zofunika anafuna zochizira matenda a mitima. Ichi ndi chifukwa chakuti anati mankhwala ndi wothandizila cardioprotective.
Iwo ayenera kukumbukira kuti mankhwala amaloledwa kugwiritsidwa ntchito imodzi ndi mankhwala amene anatumidwa ku chithandizo choyenera kwa chiwindi etiology.
M'maso "Thiotriazoline" awerenge amayi apakati ndi pa mkaka wa m'mawere. Tiyeneranso ananena kuti mawonekedwe a mankhwala anati saloledwa ntchito molumikizana ndi njira zina zachipatala.
Mowa ndi Mankhwala "Tiatriazolin" kulimbikitsa kuchitapo kanthu wina ndi mzake. Pa nkhani imeneyi, ntchito zawo concomitant ndikoletsedwa.
Kusamala
The zikuchokera zikuphatikizapo sucrose ankaona miyala (mu kuchuluka kwa 2.8 mg wa pa piritsi). Choncho, kwa mlingo pazipita tsiku la mankhwala akhoza ali pafupi 22,4 mg wa thunthu. Zimenezi ayenera kudziwa odwala, odwala ndi shuga.
The njira ndi nthawi yosungirako
Mwamtheradi uliwonse "Tiatriazolin" mankhwala ayenera kutetezedwa kuwala ndi ana sangawapeze pa kutentha madigiri kwa 14 26. Alumali moyo wa mankhwala ndi zaka 3.
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