ThanziKukonzekera

"Simvastatin": ndemanga, zikuonetsa ntchito, mtengo ndi analogues

N'chifukwa chiyani ndikufunika mankhwala "Simvastatin"? Umboni za mankhwala Adzaperekedwa patsogolo pang'ono. Ifenso kukuuzani mankhwala akupezeka mu mawonekedwe umene ali zizindikiro, mavuto ndi contraindications Anzawo, momwe ndalama, mmene ayenera bwino ntchito ndi zina zotero. D.

Kenaka, Mafotokozedwe mawonekedwe ndi zikuchokera

Mankhwala "Simvastatin" akupita pa malonda mu mawonekedwe a mapiritsi. Ali wozungulira biconvex mawonekedwe ndi chizindikiro pa dzanja limodzi, komanso woyera. mapiritsi TACHIMATA, mapale otere ali 10 mg wa simvastatin. Komanso medicament zikuphatikizapo zigawo wothandiza butylhydroxyanisole, lactose, mankhwala enaake a stearate, wowuma prozhelatinizirovannogo, talc, ndi microcrystalline mapadi.

Mu phukusi, mukhoza kugula mankhwala "Simvastatin"? Zikuonetsa ntchito ya ndalama zafotokozeredwa malangizo amene ali paketi makatoni. Palinso anayikidwa ndi matuza awiri ndi miyala (zidutswa 10).

zotsatira pharmacological

Kodi mankhwala "Simvastatin"? Akatswiri alendo akusonyeza kuti zamadzimadzi-kutsitsa mankhwala izi. Chifukwa amapangidwa synthetically.

Ankaona wothandizila ndi wofooka lactone. Anthu, ndi hydrolyzed, ndipo kenako ndipamene hydroxy-asidi otumphukira.

Ntchito ya mankhwala sayambitsa kudzikundikira poizoni. Izo mofulumira zimapukusidwa ndi kumatanthauza njira zambiri synthesizing.

The katundu wa mankhwala

Kodi katundu wa mankhwala "Simvastatin"? Reviews amanena kuti chida ichi kumathandiza kuchepetsa milingo plasma wa triglycerides, okwana mafuta ndi otsika kachulukidwe lipoprotein.

Zotsatira achire pambuyo inu mumayamba kutenga mankhwala amapezeka mkati mwa milungu iwiri. The kanthu za mankhwala akhala wosasunthika pa nthawi yonse ya mankhwala. Pambuyo kulipira mapiritsi mafuta mlingo pang'onopang'ono akubwereranso ku ntchito koyamba.

Pharmacokinetics

mankhwala "Simvastatin" yaitali bwanji odzipereka? Akatswiri Mlendo kuti mayamwidwe ndalama ndi mkulu. Atalandira mankhwala mu ndende ake apamwamba mu magazi kukufika pambuyo maola 1.5-3 ndi yafupika 90% pambuyo pa 12 maola. Kulankhulana ndi madzi pafupifupi 95%.

Kagayidwe wa mankhwala chiwindi. Theka moyo wa metabolites ndi maola pafupifupi awiri.

Anasonyeza medicament ndi ndowe komanso kudzera impso.

Mankhwala "Simvastatin": zikuonetsa ntchito

Ndalama analimbikitsa ntchito hypercholesterolemia, ndi matenda a mitima. Mankhwala mankhwala amenewa ayenera kukhala dokotala ndikatha kumfunsafunsa dokotala.

Choncho Mulimonsemo mukhoza kutenga miyala "Simvastatin"? Kuchokera pa zimene zikutanthauza akapatsidwa? Malinga ndi malangizo, mankhwala tikulimbikitsidwa pamene:

  • hypercholesterolemia chachikulu;
  • kupanda a zakudya ndi otsika mafuta chakudya ndi njira zina sanali mankhwala (kuwonda, masewera olimbitsa thupi) odwala ndi atherosclerosis inatsekeratu;
  • ophatikizana hypertriglyceridemia ndi hypercholesterolemia, amene sitisintha katundu thupi ndi kudya zakudya zapadera.

Kodi zina zotchulidwa mankhwala "Simvastatin"? Zikuonetsa ntchito chida ino pakali pano:

  • kupewa m'mnyewa wamtima infarction;
  • kuchepetsa chiopsezo cha matenda a mtima (mwachitsanzo, chosakhalitsa ischemic kapena matenda opha ziwalo);
  • retardation a atherosclerosis m'zotengera inatsekeratu.

contraindications

Tsopano inu mukudziwa zomwe Mankhwala "Simvastatin". Zikuonetsa ntchito chida akhala anapereka pamwamba. Komabe, mankhwala pali contraindications. The chikhalidwe zotsatirazi likukhudza kuti:

  • matenda minofu (kapena otchedwa myopathy);
  • chiwindi matenda zikuchitika mu gawo yogwira;
  • zaka 18;
  • kulimbikira kukwezedwa kwa michere chiwindi (kuphatikizapo etiology osadziwika);
  • hypersensitivity kuti mankhwala kapena zigawo zake payekha (kuphatikizapo tsankho lactose);
  • hypersensitivity kuti njira zina statin zino.

Mosamala yokonza phwando

Medicament "Simvastatin", mtengo wa chomwe chili m'munsimu, ndi chisamaliro makamaka anapatsidwa odwala amene amamwa mowa mwauchidakwa, komanso anthu awa limba kupatsidwa zina (ndi mankhwala immunosuppressive).

Komanso, nkhani kumabweretsa mosamala anatengedwa mu zinthu wopita ku chitukuko cha kulephera aimpso (mwachitsanzo, hypotension, matenda pachimake zachilengedwe opatsirana, yafupika, kapena M'malo mwake, kochulukira tonus minofu minofu, anasonyeza kagayidwe kachakudya ndi endocrine matenda, khunyu, zipolowe electrolyte bwino, opaleshoni, kuphatikizapo mano ndi zoopsa).

Mankhwala "Simvastatin": ntchito ndi mlingo

Akuti isanafike kuyambitsa mankhwala zikutanthauza wodwala ayenera kukumana ndi muyezo hypolipidemic zakudya. Zodabwitsa ndizakuti, tiyenera kutsata mu njira ya mankhwala.

"Simvastatin" piritsi kutumikiridwa kamodzi tsiku lililonse madzulo. Ngakhale kumwa mankhwala ayenera sizigwirizana ndi kumwa chakudya.

Analimbikitsa Mlingo wa mankhwala a hypercholesterolemia ndi 10-80 mg wa pa tsiku.

kusintha mlingo ayenera ikuchitika pa intervals pamwezi. Choyamba, wodwala ayenera kutenga 10 mg, ndiye 20, 30 ndi zina zotero. D. Nthawi zambiri mulingo woyenera achire zotsatira analandira pamene kulandira 20 mg wa mankhwala.

Mlingo wa mankhwala zimadalira m'badwo wodwala matenda ake ndi zina zotero. Pa nkhani imeneyi, monga mankhwala kukhala akapitawo dokotala, atafufuza mtima ndi kuona zachipatala.

zosiyanasiyana chokhwima

Mofanana ndi mankhwala osokoneza bongo, medicament "simvastatin" alinso mavuto. Pakati ambiri ali zotsatirazi:

  • M'mimba ululu, matenda a chiwindi, kudzimbidwa, kapamba, flatulence, kusanza, anakwezedwa chiwindi michere, kutsekula m'mimba, ndiponso nseru.
  • Asthenic syndrome, mkhutu tanthauzo la kukoma, mutu, kusawona bwino, chizungulire, neuropathy zotumphukira tulo, paresthesia, omangana minofu.
  • Angioedema, eosinophilia, polymyalgia rheumatica, urticaria, lupus-monga matenda, vasculitis, dyspnea, thrombocytopenia, amamva, kuchuluka erythrocyte sedimentation mlingo, ankatenthetsa wa khungu, malungo, photosensitivity, nyamakazi.
  • Ziwengo, alopecia, dermatomyositis, kuyabwa.
  • omangana Myopathy, rhabdomyolysis, myalgia, kufooka, minofu.
  • Magazi m'thupi, yafupika potency, mtima, aimpso kulephera (pachimake).

malangizo Special kulandira medicament

Musanagwiritse ntchito mankhwala muyenera kuwerenga malangizo mosamala. Lembali limati:

  • isanayambe mankhwala n'kofunika phunziro la chiwindi;
  • mankhwala "Simvastatin" sayenera kumwedwa ngati kulephera aimpso ndi chiopsezo rhabdomyolysis adakula;
  • mankhwala akhoza kukhala mavuto pa mwana wosabadwayo;
  • Iwo ali osavomerezeka kutenga mankhwala kuti akazi wobereka zaka amene sagwiritsa ntchito njira za kulera zosiyanasiyanazi;
  • Pa mankhwala sayenera nkhanza mowa;
  • pamene mankhwala wodwala ayenera kutsatira zakudya hypolipidemic;
  • munthawi yomweyo phwando madzi manyumwa umathandiza mlingo wa kukula kwa machitachita mbali;
  • kukonzekera zingakhale zothandiza ngati monotherapy, ndipo pamodzi ndi ntchito sequestrants ya ndulu acid.

Analogs ndi mtengo wa mankhwala

Tsopano inu mukudziwa kuti ndi mankhwala "Simvastatin". Analogues, mtengo wa mankhwala uno udzaperekedwa tsopano.

Ngati ndi ntchito yosatheka zikutanthauza akhoza m'malo ndi mankhwala ena monga "Simvakard", "Avestatin", "Holvasim", "Aktalipid", "Sinkard", "Aterostat", "Simplakor", "Vasilip", "Simli" "Vero -Simvastatin "," Simgal "," Zovatin "," Simvor "," Zocor "," Simvastol "," Zorstat "," Simvalimit "," Ovenkor "," Simvakol "," Simvageksal "ndipo T. d.

mankhwala Price "Simvastatin" si mkulu kwambiri ndipo watsala 240 rubles kwa mapiritsi 20.

Reviews a medicament

odwala ambiri kale "Simvastatin" mapiritsi, onani Mwachangu ake okwezeka. The mankhwala ndi mofulumira Sachita mafuta m'thupi, kuteteza chitukuko cha matenda osiyanasiyana.

Komabe, odwala ena ndi wosasangalala wodutsapo mankhwala mafuta mlingo adzawuka kachiwiri ndi zimadza ndi m'mene ziriri pano ndi.

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