Thanzi, Kukonzekera
"Buspirone": ndemanga, malangizo ntchito, analogs
"Buspirone" amatanthauza ndalama zomwe zimakhudza wamanjenje dongosolo. Ndi anxiolytic, cholinga kuthetsa nkhawa ndi mantha, normalization wa tulo, kusintha bwino pamaso pa gwero lachisokonezo. Miyala "Buspirone" ena contraindications, ndipo angathe kuyambitsa zotsatira zoyipa.
Kapangidwe ndi mawonekedwe a "Buspirone" mankhwala
The mankhwala ndi alembedwe piritsi pa mlingo wa 5, 10 ndi 20 mg. The yogwira mankhwala mankhwala - buspirone. Wothandiza zinthu monga hydroxide potassium wowuma chimanga, magnesium stearate.
zotsatira pharmacological
Ntchito ya sedative mankhwala, anxiolytic. mankhwala kuthetsa zizindikiro za mantha a vegetative ndi maganizo. zikutanthauza limagwirira a kanthu n'komwe, koma amadziwika kuti "Buspirone" chosiyana ndi benzodiazepines ndi mankhwala ena anxiolytic kwenikweni.
A amphamvu ochepetsera amasintha CNS pambuyo polandira olumikizidwa ku makina "buspirone" miyala. Malangizo ntchito limasonyeza kuti mankhwala amachepetsa mapangidwe ndi kutulutsidwa serotonin, kubweza serotonergic, kumalimbikitsa kutsekereza dopamine D2-maselo (postsynaptic ndi presynaptic malo), Iyamba malemeredwe wa manyuroni dopamine ili mu midbrain lapansi. Pambuyo chiyembekezo chakuti mankhwala ali mwaonapo pakutchulidwa cha mavuto obwera ndi nkhawa kubwerera.
mankhwala cholinga cha utsogoleli m'kamwa. Ozama mu thupi mu nthawi yochepa iye kuganizira thirakiti m'mimba. Chifukwa, kagayidwe kwambiri bioavailability ndi 4%. Mlingo pazipita mankhwala m'magazi kukufika ola limodzi pambuyo malowedwe mu kapepala kakuti m'mimba. Theka moyo ikuchitika kwa maola 2-3, kumanga kwa mapulotini plasma limafanana ndi 95%. Wopitiriza ntchito "buspirone" sikumangotikhudza nchito zake.
Pa mankhwala, kodi si monga kuyembekezera "Buspirone" amatanthauza kwenikweni. Malangizo ntchito zimasonyeza kuti mphamvu ya mankhwala ndi nthawi kuchokera 7 mpaka tsiku la 14 la anavomereza. Zotsatira pazipita mankhwala akuwonetseredwa masiku pafupifupi 120 mankhwala.
Zikuonetsa "buspirone"
Akatswiri mankhwala pamene kumverera ngozi, kuwulula mantha ndi nkhawa, ayi chinachititsa irritability zikuchitika gwero lachisokonezo ndi kugona matenda wachete, ndi khalidwe ndi mwadongosolo. mankhwala ndi oyenera zochizira matenda somatic, vegetative dystonia ndi maganizo, kuthetsa nkhawa, achire mowa.
Contraindications kulandira "Buspirone" mankhwala
"Buspirone" (analogues wa mankhwala komanso) ali contraindications. Mankhwala choyambirira amaletsedwa kujambula mu Zikatero:
- khungu (chatsekedwa mtundu);
- lolemera njira pathological kunachitika chiwindi ndi impso;
- khunyu;
- matenda a mtima, mavuto ndi mitsempha;
- zotupa pa mundawo kupuma;
- myasthenia gravis;
- Hypersensitivity kwa zigawo zikuluzikulu;
- nthawi wobereka, akumuyamwitsa pamtima;
- zaka zosakwana zaka 18.
Ngati pali kutiletsa mankhwala mankhwala kuti wodwala "Buspirone" mbiriyakale ya khunyu kapena khunyu.
Asanayambe mankhwala ayenera kuonanso tilinazo wodwalayo kwa mankhwala.
Kugwiritsa ntchito ndalama, mlingo
Pa mankhwala amatanthauza "buspirone" ntchito za miyala mogwirizana ndi malangizo a dokotala amachitira. kalozera Official lili ndi mfundo zimene zimafunika kuti mlingo uliwonse mtima osiyana, mwachitsanzo. K. aliyense chithandizo dera Mzimuyo mphamvu ya mankhwala anachita. Mlingo zimadalira thanzi wodwalayo. ayamikira General ali motere:
- Koyamba siteji - 3 Mlingo wa 5 mg wa mankhwala;
- kupitiriza mankhwala - kuwonjezeka pang'onopang'ono mlingo kugwilizana ndi imeneyi ya masiku 2-3 (ngati pali kufunika);
- yopereka kwa mlingo pazipita tsiku la 50 mg (pakalibe zotsatira anakhumba).
Miyala "Buspirone" malangizo ntchito zilolezo kokha kutenga maonekedwe a lonse, iwo sangakhoze zidzasungunuka mu madzi, akupera ndi kutafuna. Mankhwalawa ndi kuledzera ndi ndalama mvula ya madzi, pamene amwedwa pa nthawi iliyonse tsiku payekhapayekha kudya chakudya. Kutalika kwa mlingo analimbikitsa ndi miyezi 4. Motalikira nthawi imeneyi ankachitira "buspirone" ali osavomerezeka.
Zotsatira zoyipa "buspirone"
Pamene mankhwala ena zochita oipa lake angathe kuonedwa. Mwachitsanzo, kugona, kuwonongeka ambiri thanzi, kufooka, kutopa, mphwayi. Ngati pali zotsatira amenewa amafuna kuchotsa mankhwala. Lankhulani ndi dokotala wanu ndipo anamuuza za kusintha zoipa m'thupi pambuyo kutenga mankhwala "Buspirone". Malangizo ntchito Zikatero Ndi bwino kuchepetsa mlingo wa wothandizila. Ngati mavuto sapita kwina, dotolo ali m'malo mankhwala ena mankhwala yoyenera kwambiri.
Nthawi zina kwambiri, kugwiritsa ntchito "buspirone" zimabweretsa chisokonezo dongosolo m'mimba. Mwachitsanzo, pangakhale kunyansidwa ndi kutentha, kenako anayamba kusanza. N'zotheka ululu m'dera epigastric. Pangakhale zotsatira zina zoyipa. Zizindikiro zonse izi kusonyeza tsankho mwa zigawo mankhwala.
Ambiri osokoneza "Buspirone" mankhwala
Ngati chida ntchito pa mlingo waukulu kuposa osavomerezeka, munthu akhoza kuona zizindikiro za mankhwala osokoneza bongo. Zikuphatikizapo kunyansidwa ndi kusanza, kusokonezeka m'mimba mwa mtundu wina. The chizungulire mtima, kuchepetsa ana, akhoza kukhala imfa mwachidule kutsitsimuka. Odwala kusiya review mankhwala amatanthauza "Buspirone Sandoz" anati kuthekera chisokonezo, chapamwamba nthambi kugwedeza. Pakati pa zinthu zina cha mankhwala osokoneza bongo - irritability, irritability, kusintha kawirikawiri maganizo. Overdosing amaliona ndi lavage chapamimba, utsogoleli wa adamulowetsa mpweya mu thupi, mankhwala symptomatic ndi kuchititsa kulamulira zonse magazi, kugunda kwa mtima, ntchito kupuma. adakalibe lenileni la mpumulo zizindikiro cha mankhwala osokoneza bongo "buspirone" kulibe. Dialysis m'mavuto oterewa wosatenga zotsatira ankafuna.
Mogwirizana ndi zinthu zosiyanasiyana ndi mankhwala ena
Nthawi zina pamene kuphatikiza zoletsedwa mankhwala ena mankhwala "Buspirone" malangizo ntchito analogues tilingalire mmalo mwa malo pachiyambi. Amadziwika kuti mankhwala sayenera kumwedwa nthawi imodzi ndi asamakhale ndi nkhawa, mankhwala chifukwa patsogolo zotsatira za mankhwala atengedwa. Mankhwalawa "buspirone" koyenera kuti achotse kumwa mowa. Simungathe kuphatikiza mankhwala ndi Mao zoletsa chifukwa cha ngozi ya mavuto hypertensive.
Pamene inu kugwiritsa ntchito "Haloperidol" ndi "buspirone" m'magazi kumawonjezera mlingo wa mankhwala. Yonseyi mankhwala ndi "trazodone" amatsogolera kuwonjezeka kwambiri alt.
Chifukwa cha zinthu zatsopano zokhudza nyama, kungasokoneze lake sanali wapezeka pa mankhwala. Komabe, pofuna kupewa zochita oipa thupi kuvomereza ndi kupeleka.
"Buspirone" malangizo ntchito ndi ngati chida amene kagayidwe mu chiwindi. Mu ndondomekoyi nawo CYP3A4, pokhala isoenzyme zikuthandiza processing chamoyo kukonzekera. Pachifukwa ichi, mogwirizana ndi kumachitika "buspirone" ndi mankhwala amene ali inducers, kapena zoletsa cha enzyme ndi.
Features ntchito mankhwala
Ngati, pamene mkaka wa m'mawere, pali kufunika mankhwala zochokera phwando "buspirone" yoyamwitsa mongoyembekezera ndinayima.
Pali zoletsa zina pamene kusokonezeka kwa ntchito kwa ziwalo. Mwachitsanzo, ngati muli ndi vuto la chiwindi ayenera kusamala nthawi chithandizo ndi zonse kuwunika kusintha komwe kumachitika ndi thanzi. Contraindications yekha aakulu kuvutika mu kugwira ntchito kwa thupi. N'chimodzimodzinso ndi ntchito ya impso.
Ponena za poika wothandizira ku opanga osiyana, Vol. H. "Buspirone Sandoz" mankhwala, ndemanga mankhwala akusonyeza kufunika kulemekeza malamulo. Kulemba mankhwala, katswiri ayenera kudziwa kuti chida ichi si okhoza kuthetsa kusiya zizindikiro chifukwa benzodiazepine, ndi cholinga chake zoterezi sizingatheke ngati si phasing mwa mankhwala anxiolytic anapangidwa pamaso chithandizocho.
Odwala ayenera kudziwa kuti mapilisi "Buspirone" zingakhudze chisamaliro, makamaka pachiyambi cha mankhwala, choncho ndi bwino kuti mongoyembekezera kupewa zinthu zokhudza udindo wapadera ndi kuchuluka ndende. Ena ntchito kungakhale zikanavulaza thanzi.
Pankhani chithandizocho "Buspirone" njira, madokotala zenizeni za mankhwala makamaka positive. Komabe, akatswiri amanena kuti m'pofunika perekani molondola yekha ndi zizindikiro yoyenera ndiponso Mlingo mulingo woyenera. Tikumbukenso kuti mavuto kuti kuwuka kwa okhazikika kungasokoneze pampanipani tsiku ndi tsiku, mankhwala ndi anxiolytics zambiri Sikuti.
Kulandira kutanthauza odwala "buspirone" ndi mlingo wosiyana, mwachitsanzo mankhwala "buspirone 10 mg" mavoti zikuimira ntchito njira. Anthu amene ankapatsidwa mankhwala, onani kuti dokotalayo anawachenjeza kuti kugwiritsira ntchito bwino mankhwala ena, monga kulera m'kamwa, mankhwala matenda a shuga n'lakuti olimbana kuchepetsa kuthamanga kwa magazi, mankhwala kuthetsa maganizo ndi mankhwala monga glycosides mtima , neuroleptics.
Aimpso kulephera ndi woopsa matenda enaake chiwindi amafuna kuchepetsa mayunitsi mlingo. Mu milandu, njira "Buspirone Sandoz" amakambirana mmene anthu pofotokoza mankhwala chofunika zimene tikubweretsazi kuyang'aniridwa ndi dokotala. Akunena za kusintha pang'ono thanzi.
Odwala ndi mankhwala khunyu konse Kwalamulidwa chifukwa chiopsezo khunyu. zochiritsira zamtunduwu odwala awa ndi woopsa kwambiri ndipo iyenera kuchitidwa ndi kugwiritsa ntchito mankhwala ena. Odwala amene amakonda nkhanza mankhwala ndipo ndi mbiri kudalira mankhwala ayenera kulandira chithandizo kuyang'aniridwa okhwima katswiri (liwuli malingana "buspirone" sanali).
Kafukufuku wasonyeza kuti "Buspirone" pambuyo masabata 3-4 mankhwala pamene Alamu si ogwira, choncho palibe lingaliro kuwachitira kwa nthawi yaitali. Chifukwa chosowa mauthenga pa chitetezo mankhwala kwa ana a udindo wake sakhala ndi anthu osakwana zaka 18 zakubadwa.
Chithandizo cha mitundu yosiyanasiyana ya mankhwala ndi mankhwala "Buspirone hexane" amakambirana akatswiri ena mmene osamveka mankhwala chifukwa kugona mavuto, zikamera wa irritability ndi nkhawa nthawi zina chizindikiro cha matenda aakulu psychomotor.
Analogs, ndemanga za mankhwala "Buspirone"
M'malo mankhwala analogi ziyenela kuchitidwa pambuyo kupeza malangizo dokotala. Pali m'malo abwino kwa mankhwala, "Buspirone" - "Spitomin". Umboni bwanji kuti ntchito yake ndi ofanana ndi zochita za ndalama pachiyambi. "Spitomin" ntchito zochizira zinthu amene limaleka ndi "Buspirone". Reviews zabwino, choncho ngati mukufuna n'zotheka kuti agwiritse ntchito mmalo izi, koma atakambilana ndi katswiri. A kuchita chimodzimodzi zimatheka chifukwa kukhalapo kwa yemweyo yogwira pophika. The yabwino kwambiri "Spitomin" awonetsera mu chithandizo cha odwala matenda nkhawa.
Pambuyo mankhwala ndi "Buspirone" umboni ungachoke osiyana, koma kwenikweni chifukwa cha zimenezi ndi zabwino. Kodi anatsimikizira nchito zake? Reviews madokotala akusonyeza kuti mankhwala ndi yogwira hydrochloride pophika buspirone ali bwinobwino kumenyana mawonetseredwe nkhawa zosiyanasiyana mwamphamvu ndi chiyambi, koma zotsatira zake kamodzi pafupifupi padera, akhoza amangoona patapita nthawi yina, ndicho - pambuyo mlungu umodzi kapena iwiri. Kuwona pazipita zotheka achire zotsatira, amafunabe mankhwala kwa mwezi umodzi.
"Buspirone" amalandira mayankho abwino odwala milandu kumene kunali zotsatira palibe mbali, ndi mankhwala lake anakumana chabwino. Nthawi zina padzakhala anachita zoipa lake, koma kawirikawiri pamene thupi Kodi simuzindikira zigawo zikuluzikulu za mankhwala. Kuyambira ndemanga, inali kudziŵika kuti mankhwala akhoza limodzi ndi misala ndi ntchito sotsioterapevticheskimi. Nthawi zina odwala ndi m'mimba chowawa zochita, chizungulire ndi kufooka. Ambiri osokoneza - chodabwitsa osowa.
Motero, ntchito mankhwala "Buspirone" mayankho odwala ankachitira N'zoona kuti nthawi zambiri kusiya mfundo za zotsatira zina zoyipa. Maphunzirowa zikhazikitsidwe makhalidwe munthu wa thupi la munthu, thanzi lake, ndi mulingo woyenera kwambiri mlingo lililonse. Ngakhale kulamulira zonse dokotala, wodwalayo ali wofunikila kuwerenga malangizo musanayambe chithandizo.
"Buspirone" - mankhwala si kawirikawiri kungathandize kuti apange mavuto ndi ambiri osokoneza, si osokoneza panachitika zoipa pambuyo Kulipira ake, ndipo nthawi zambiri amachita ntchito yake.
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