Thanzi, Kukonzekera
"Tolperisone": analogues, mtengo, malangizo ntchito
Matenda okhudza dongosolo minofu ndi mafupa kumachitika kuphipha minofu ndi kuwonjezera kamvekedwe. Odwala amene ali okhumudwa, chithandizo chokwanira zochokera ntchito relaxants minofu. Madokotala amakonda kulemba "tolperisone." Analogues, mtengo, malangizo ntchito mankhwala tidzakambirana m'nkhani.
Medicament ndi yogwira hydrochloride mankhwala tolperisone alipo mapiritsi. The medicament zina anawonjezera asidi stearic ndi citric acid, komanso lactose ndi crospovidone.
zotsatira pharmacological
"Tolperisone" analogues mankhwala ndi relaxants minofu, ndi kanthu chapakati. Limagwirira cha mphamvu ya mankhwala pa thupi asanamvetsetse.
"Tolperisone" amatipatsa mankhwala oletsa ululu pamalopo. Amadziwika kuti medicament chifukwa cha mankhwala yogwira alipo zikuchokera, kumatha hypertonus minofu, kuchititsa ululu kusiyiratu. Mankhwala bwino kufalitsa zotumphukira, antispasmodic ndi kukwaniritsa adrenoceptor kutsekereza zotsatira, izo kumabwezera mmbuyo ntchito ya gawo caudal wa ku reticular mapangidwe a ubongo.
"Tolperisone" analogues, ofanana matanthauzo angathe kuchotsa gipertonus striated spasms minofu ndi kuthetsa mu zochitika zonsezi pamene mavuto anayamba chifukwa kuwononga matenda mtima kapena entsefalopapii.
Kuti mankhwala mankhwala "tolperisone"?
Madokotala mankhwala mankhwala "tolperisone" pamaso pa nkhani zotsatirazi:
- matenda limodzi ndi akulu kuphipha, monga sitiroko, mwiniwakeyo sclerosis; mwa matenda amenewa - encephalomyelitis, myelopathy;
- matenda, zomwe ndi mawonetseredwe a akulu dystonia; zikuphatikizapo oziziritsa ziwalo, zina encephalopathy;
- njira chifukwa cha zimene zinkakhala dongosolo minofu ndi mafupa, pali olemba minofu spasms; Zikuphatikizapo nyamakazi zokhudza mfundo yaikulu, ndipo lumbago; Zizindikiro ngati spondylarthritis, spondylitis.
Pamene ntchito kuipidwa "Tolperisone" analogs ntchito pofuna kuchiza acrocyanosis, arteriosclerosis, matenda Raynaud a, angiopathy.
Contraindications kulandira "tolperisone"
mankhwala si Kwalamulidwa kwa anthu pansi zaka 18, odwala myasthenia gravis, akazi adzabala mwana ndi wozengereza yoyamwitsa, odwala amene sangakhoze kulekerera lactose ndi mbali zina lokonzekera.
Buku lili zofooka. Mankhwalawa odwala ndi opuwala chiwindi ntchito ndi impso mankhwala kugwiritsidwa ntchito mosamala kwambiri.
Nthawi zina "tolperisone" analogues yoikidwa pa mimba. Koma popeza zotsatira za mankhwala pa thupi la amayi apakati sichinayambe kuphunzira, ntchito zawo n'chotheka pa nthawi imene phindu kwa thupi la mkaziyo ali wamkulu kuposa chiopsezo kwa mwana wosabadwayo. mankhwala chithandizo pa trimester amafuna kusamalidwa kuti boma la thupi la wodwalayo. Mu mankhwala "tolperisone" yoyamwitsa mongoyembekezera ndinayima.
Kugwiritsa "tolperisone": Mlingo
medicament The cholinga ntchito mkati pambuyo kumwa chakudya (piritsi anatengedwa pa chopanda kanthu m'mimba ali otsika bioavailability). Analimbikitsa mlingo chithandizo koyamba 50 mg wa mankhwala 3 zina tsiku lililonse. M'kupita kwa nthawi, chinawonjezeka 150 mg, koma osati zikuchepa, koma pang'onopang'ono. Pafupipafupi mankhwala akhala sichinasinthe. Kutalika kwa mankhwala kwa wodwala aliyense anatsimikiza payekha.
The mankhwala ndi mankhwala yogwira pansi pa dzina la tolperisone hydrochloride, analogs mankhwalawa odwala ndi chisokonezo anamuona pa chiwindi ndi impso (zikutanthauza kuunika) ntchito mosamala kwambiri ndi kuwasankha Mlingo. Pali kufunika polojekiti zonse odetsedwa thanzi. matenda aakulu ndi contraindication kugwiritsa ntchito "tolperisone."
zotsatira zoyipazi
A ambiri ndemanga zikuonetsa tolerability wabwino wa zigawo zikuluzikulu ya zinthu alipo zikuchokera mankhwala. Development mosiyanasiyana chowawa pambuyo kutenga mankhwala si makamaka wamba. kawirikawiri, pali kufooka m'minofu, nthawizina pali mutu, ndi kukhalapo kwa matenda oopsa. wosokoneza mu makhalidwe matumbo, imene pali kunyansidwa ndi kusanza. Ku thupi lawo siligwirizana akhoza kupezeka angioedema, pruritus, urticaria mutadya "Tolperisone" kukonzekera. Zotsatira zake zoyipa komanso ndi analogues.
ambiri osokoneza
No milandu cha mankhwala osokoneza bongo zalembedwa. Chifukwa cha kutenga mlingo woposa analimbikitsa, angathe hypotension, nkotheka kuyan'anila za kupuma ndi ntchito mtima. Kuthetsa ngati mawonetseredwe zofunika chapamimba lavage ndi kukhazikitsa chithandizo (wothandiza, symptomatic).
mogwirizana mankhwala "tolperisone"
Ngati mankhwala ntchito ndi asidi niflumic, anthu amamuona kuti zotsatira zake. "Tolperisone" Komanso kumawonjezera ntchito "clonidine", mankhwala psychotropic, mankhwala kupereka mankhwala oletsa ululu ndi minofu zotumphukira relaxants.
"Tolperisone" analogues akhoza pamodzi ndi mankhwala ena - mankhwala, kuphatikizapo Mowa, mitsempha, ogonetsa.
Pamene pamodzi ndi minofu ena relaxants kanthu yemweyo amene anawamasulira kuti "Tolperisone" mapiritsi, amafuna kungachepetse mlingo wa wothandizila lapansi.
Mankhwala zingakhudze mankhwala kagayidwe wa CYP2D6 isoenzyme nawo, kuwonjezeka maganizo awo.
Analogs, mtengo wa mankhwala
Kodi m'malo "tolperisone"? A zabwino ndi otchuka kwambiri mankhwala ndi "Mydocalm", ngati kuli kofunikira angagwiritsidwe ntchito m'malo yemweyo chigawo yogwira.
Mumadziwika mankhwala embodiments ena, monga "tizanidine" ndi "Sirdalud". Kuwonjezera zida izi, mukhoza kugwiritsa ntchito "Tizaludom", "Tizanilom", "Liorezalom" kapena "Baklosanom". Pali wogwirizira wina - "tolperisone-OBL». mankhwala ndi otsika mtengo kuposa amagwiritsidwa ntchito "Mydocalm", yemwe ali mmodzi wa anthu otchuka analogues mankhwala "tolperisone." Price, analogues - maziko kusankha kwambiri opindulitsa ndi ogwira mmalo.
Odwala amene ankapatsidwa minofu anasiya "tolperisone" kwenikweni okhutitsidwa ndi zotsatira zake. Mwachangu Wamkulukulu amatchuka kuthetsa spondylosis ndi spondylarthritis, mankhwala, ngati n'koyenera, encephalomyelitis, mwiniwakeyo sclerosis. Mtengo pafupifupi miyala ndi mlingo wa 50 mg wa opaka 140, ndi mlingo wa 150 mg -. 190 rubles.
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