Thanzi, Kukonzekera
"Omeprazole" kapena "Ultop" - umene uli bwino? Kufotokozera za mankhwala, zizindikiro ndi contraindications, mitengo
Mankhwala a zotupa anam'peza wa mucosa m'mimba kapena kapepala m'mimba ambiri - kuipidwa ndi yaitali ndondomeko. Ichi ndi chifukwa osati chakuti acid amathiridwa, mbali ya madzi chapamimba, umachuluka pang'onopang'ono mucosa chilema, chosinkhasinkha zimakhala yekha, koma kugwirizana ndi pamaso pa matenda Helicobacter pylori bakiteriya. Pofuna kupewa kufalikira kwa chilema ndi atsogolere kuchira mofulumira akudwala, madokotala mankhwala "omeprazole" kapena "Ultop". Chabwino n'chiti, tikambirana chiyani m'nkhani ino.
limagwirira kanthu
Ngakhale kuti mankhwala ali ndi dzina zosiyanasiyana yogwira pophika mu chinthu chomwecho - omeprazole. Amene ndimachiza ndi mankhwalawa?
Malinga ndi makhalidwe mankhwala mankhwala pafupifupi insoluble m'madzi, koma sungunuka kwambiri Mowa kapena methanol.
Zochita matenda, omeprazole ntchito zikuchokera mankhwala osiyanasiyana, kuphatikizapo osakaniza, monga wothandizira kwa zilonda zam'mimba. "Omeprazole" kapena "Ultop" - umene uli bwino? Nthawi zambiri ndimadzifunsa funso limeneli, odwala ndi madokotala.
Limagwirira cha zochita zochokera chopinga otchedwa purotoni mpope - yeniyeni zoyendera mapuloteni ili mu selo nembanemba ya maselo secretory m'mimba. Ndi kuchepetsa kuvomera ayoni wa hydrogen mu cytoplasm ya maselo amenewa secretory utachepa zopanda amabala acid amathiridwa ndi acidity wa amachepetsa chapamimba madzi, imbaenda kuchepetsa kuwonongedwa minofu ndi amakonda machiritso mofulumira zilonda.
Pharmacokinetics
Omeprazole bwino kumabwezera mmbuyo onse analimbikitsa ndi woyambira yopanga acid amathiridwa pa mlingo chomwecho yozungulira kwenikweni. Pamene limodzi m'kamwa makonzedwe a 20 mg wa "omeprazole" kapena phwando mlingo "Ultop" kukonzekera - 20 mg, acidity kuchepa zimawonedwa mu Ora loyamba, kuyambira mankhwala ndi mofulumira komanso odzipereka kwa lumen wa matumbo ndipo amabwera mu zokhudza zonse kufalitsidwa.
Ngakhale theka moyo wa formulations yogwira wothandizila ndi maola pafupifupi awiri, chopinga wa yopanga acid amathiridwa zimawonedwa mwa masiku pambuyo mlingo umodzi.
kudutsa Omeprazole analigawa ndi chiwindi ndi biliary thirakiti mucous nembanemba m'mimba, pafupifupi Kodi mkatikati kwa magazi mu ubongo chotchinga ndi kwathunthu womangidwa kwa mapulotini plasma. The digiri ya kumanga ndi yamasika kungakhale kwa 90-95%.
Excretion wa omeprazole ikuchitika makamaka mu mkodzo, ndi za 60-77% ali excreted mu mawonekedwe a metabolites monga gidroksiomeprazol acid carboxylic. Ambiri mwa conjugates chifukwa kuonetsa pafupifupi palibe ntchito antisecretory, kupatula sulfonomeprazola. Thupi otsala mbali ya thunthu mankhwala kuperekedwa ndi kachigawo m'mimba mwa ya ndulu ndi ndowe.
mwapadera ayenera pharmacokinetics wa omeprazole odwala ndi insufficiency kwa chiwindi. Ndi kuchepetsa kagayidwe mankhwala kufika bioavailability pazipita ndi nthawi theka moyo yaitali maola atatu. Odwala ndi insufficiency aakulu aimpso kubweza excretion wa metabolites wa omeprazole monga mwa mayeretsedwe wa madzi a m'magazi creatinine.
zikuonetsa
Mankhwala "omeprazole" ndi "Ultop" anasonyeza ntchito pa zilonda zam'mimba zilonda za m'mimba thirakiti, limati hyperacidity (kuphatikizapo gastritis), syndrome Zollinger-Ellison zinthu postoperative matenda Reflux. Mankhwalawa akhoza akulimbikitsidwa mankhwalawa si chilonda dyspepsia Genesis mankhwalawa mavuto chifukwa cha sanali steroidal mankhwala mankhwala protivovospalitelnymim (analgesics, antipyretic), komanso zochizira wopepuka kutentha amenewa amapezeka zosaposa 2 nthawi pasabata.
Ngakhale malangizo mu zikuonetsa ntchito mankhwala "Omeprazole" kuti amachitira mankhwala, amadziwa zokha katswiri ophunzitsidwa. Choncho, ngati mukuona akudwala, kwa mundawo m'mimba, muyenera kupita ku chipatala ndipo osati kudzimvera medicate.
contraindications
mitundu yonse ya mankhwala, kuphatikizapo miyala "Omeprazole" ali contraindicated mu kukhalapo kwa odwala hypersensitivity kuti mankhwala, komanso ana. Kuchepetsa secretory ntchito ya m'mimba pamene limati hypoacid ndi atrophic gastritis alinso contraindication kuikidwa kwa omeprazole.
zotsatira zoyipazi
Za mankhwala "Omeprazole" ndi "Ultop" ndemanga ndinena mwa kuchepetsa asidi-kupanga ntchito ya m'mimba, ku kachigawo m'mimba ayenera kuti chifukwa kudzimbidwa, bloating, kudzimbidwa, kusanza ndi ululu m'dera epigastric. Kawirikawiri anati candidiasis, pakamwa youma, kapena chitukuko cha atrophic hypoacid gastritis, polyposis wa intestine lapansi.
Kuyambira wamanjenje dongosolo (imalandira athandizira), mungachite mutu, malaise, nkhawa ndi nkhawa, maganizo ndi mavuto a m'maganizo. N'zotheka zikamera matenda a ntchito zithunzi kuti akhoza kukhala okhazikika.
Matupi awo sagwirizana anachita omeprazole n'zochepa. Vuto zikhoza ming'oma, kuyabwa. Ndi zolemba otsika pafupipafupi gladomyshechnyh bronchial chitukuko kuphipha selo angioedema ndi kupitirira patsogolo za mtundu anaphylactic zochita ndi chitukuko cha sosotoyaniya mantha. Casuistically taonera chitukuko cha gynecomastia, maonekedwe a ululu pachifuwa.
dosing
"Omeprazole" kutenga pa chopanda kanthu m'mimba ndi madzi. Mu gulu lapadera la odwala kuona vuto Pomeza makapisozi a mankhwala. Pankhaniyi, izo tikulimbikitsidwa kutsegula kapisozi ndi nkhani zake ku slurry kuti akonze madzi ofotokoza. kuyimitsidwa ayenera osachepera theka la ola pambuyo kuphika. Mlingo tsiku, mlingo umodzi, komanso njira ya mankhwala chimaika dokotala.
Features ntchito mu mimba ndi kuyamwitsa
Data pa chitetezo cha omeprazole mu amayi apakati mulibe. Thunthu mankhwala akhoza anasonyeza kuti asapatsire. Category mmene mwana wosabadwayo sizinachitike zotsimikizika.
Ngati pali kufunika poika omeprazole panthawi yoyamwitsa, ndiye mankhwala a otsiriza ndi kukana, kuyambira mankhwala akhoza kulowa mu mkaka wa m'mawere.
Mwanjira mankhwala
Monga "omeprazole" ndi "Ultop" kuchepetsa bioavailability wa mankhwala, mayamwidwe chimene chimadalira pa acidity wa madzi muzituluka. Komanso kumabwezera mmbuyo amasulidwe mankhwala omwe kagayidwe mu chiwindi.
Kukonzekera wosabala njira jekeseni wa omeprazole akhoza ntchito maola 12 anapereka ntchito za thupi njira sodium kolorayidi ngati zosungunulira ndi maola angapo pambuyo kukonzekera pamene ntchito ngati zosungunulira dextrose njira. Ndi njira zina omeprazole si n'zogwirizana.
Ndi mankhwala concomitant mankhwala "Warfarin" ayenera kuunikira tsiku anticoagulant misinkhu mu madzi a m'magazi kapena m'njira yake kuwayang'anira ndi prothrombin nthawi.
poyizoni ndi mankhwala ambiri osokoneza
Symptomatology omeprazole ambiri osokoneza akuwonekera monga pakamwa youma, chizungulire, mutu ndi masomphenya mkhutu. Ngati poyizoni chisokonezo zotheka, pakutchulidwa kugonagona, palpitations, ankatenthetsa zotengeka.
poyizoni symptomatic mankhwala umalimbana momwe zambiri mofulumira Kupha mankhwala m'thupi. A adakalibe yeniyeni silidziŵika. Chifukwa digiri yapamwamba ya kumanga zonsezo plasma, kugwiritsa ntchito njira dialysis detoxification kosathandiza.
Kusamala
Popeza mankhwala amagwiritsidwa ntchito pofuna kuchiza zotupa anam'peza za m'mimba ndi duodenum, ndilo wothandizila etiological wa Helicobacter pylori matenda, izo akulimbikitsidwa kuthetsa tizilombo makonzedwe concomitant mankhwala antibacterial.
Musanayambe ntchito mankhwala wodwalayo ayenera kukana matenda oopsa neoplastic pa mundawo m'mimba, kuyambira Kusankhidwa "omeprazole" kungathe kubisa zizindikiro za matenda amenewa ndi kungafoole matenda oyambirira. M'pofunika kuthetsa matenda parasitic matenda, komanso kuti asa- mphamvu zinchito a chiwindi ndi impso.
"Omeprazole" kapena "Ultop" - umene uli bwino?
A bwinobwino funso ili ndi zovuta, chifukwa mankhwala yogwira, ndipo anthu awiri onsewa ndi omeprazole. Tiyeni tione mawonekedwe a amasulidwe mankhwala "Ultop". Makapisozi amapangidwa mu mlingo wa 10, 20 ndi 40 mg, komanso ufa lyophilized (40 mg wa mu botolo limodzi) kwa yokonza njira jekeseni.
"Omeprazole" zili pa msika mankhwala mu mawonekedwe a makapisozi 10, 20 ndi 40 mg wa omeprazole mu kapisozi mmodzi, komanso ufa lyophilized (40 mg wa mu botolo limodzi) kwa yokonza njira jekeseni. amaundana-zouma ufa ndi zosungunulira ndi likupezeka mu phukusi limodzi. Komanso, mankhwala zikhoza kugulidwa mu mawonekedwe a sachets (matumba ndi ufa) kwa yokonza kuyimitsidwa m'kamwa. Kawirikawiri ali "omeprazole" mapiritsi (pellets) ndi zili chomwecho wa chinthu mankhwala.
Koma ndemanga za mankhwala awa, iwo ali abwino, monga omeprazole ndi mankhwala ogwira mtima amachepetsa ntchito secretory m'mimba. The mankhwala ndi kwambiri moti ngakhale madokotala akufunsa, "bwino omeprazole Kodi" Komabe, maganizo amasiyana pakati pa anthu odwala. Kaŵirikaŵiri anachoka pa mankhwala "Ultop" ndemanga kunena za chiyambi cha kudzimbidwa pambuyo ingestion, mutu ndi nseru.
Mtengo wa mankhwala
Ndithu, mtengo wa mankhwala kudzadalira osati pa Intaneti mankhwala imene amagulitsidwa, komanso pa mtunda kuchokera mankhwala kuchipatala ndipo, ndithudi, kwa Mlengi mankhwala. Mankhwala "Ultop 'mtengo ranges ku rubles 212 kwa 360 pa paketi. The mtengo komaliza zimadalira mlingo ndipo chiwerengero cha makapisozi pa bokosi. Mankhwala "Omeprazole" mtengo uli pafupifupi kwa rubles 80 140. Mtengo chimadaliranso mlingo ndipo chiwerengero cha makapisozi pa bokosi.
Pomaliza
Only dokotala ayenera mankhwala "Omeprazole" kapena "Ultop". Mwakupambana mankhwala, akumudziwa munthu woyenera, komanso zochita zake ziyenera kuchokera pa zizindikiro ndi alili. Ziyenera adzanyamula kukumbukira kuti nthawi zambiri chinthu molimba kusankha mankhwala ndi mtengo wake.
Odwala ayenera kulabadira "omeprazole" imene ili mtengo kwambiri poyerekeza analogue "ultop". Amene ali okonzeka kulipira kwambiri, akhoza kuyang'ana kwa analogues wa mankhwala. Ngakhale angapo wapatali "Ultop" mtengo mankhwala wolungama digiri ya chiyeretso ya mankhwala, komanso zotheka zina modulating zowonjezera kukonzekera yokha.
Chirichonse chimene chinali zonse zofunika kukumbukira golide ulamuliro: kuchita musalankhule medicate. matenda oyambirira - chinsinsi chithandizo bwino!
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