Thanzi, Kukonzekera
Malangizo 'Betalok' ntchito
"Betalok" malangizo Buku limanena kuti mankhwala a pharmacological gulu beta1-adrenoceptor muzikangana. Waukulu yogwira pophika mankhwala ndi metoprolol tartrate. Chifukwa amapangidwa ndi opanga mu mawonekedwe a mapiritsi masekeli 100 mamiligalamu, ndi mmatumba mu mabotolo pulasitiki zidutswa 100 lililonse.
"Metoprolol" ali katundu pharmacological, zochokera luso la mankhwala kupereka antihypertensive ndi kanthu odana anginal. Mankhwala othandiza kuchepetsa mlingo mtima, m'mnyewa wamtima contractility ndi excitability, kumalimbikitsa deceleration njira AV-conduction. Kukonzekera "Betalok" malangizo Buku limafotokoza kuti azitithandiza kuchepetsa voliyumu mtima ndi kuchuluka kwa mpweya yochuluka myocardium lapansi. "Metoprolol" amatha kuchepetsa zotsatira za makatekolamaini pa zolimbikitsa zimakhudza awo pa mtima wodwalayo pa maganizo psycho m'thupi. Mankhwala kumakhudza hypotensive, wosasunthika pambuyo masabata awiri a mankhwala. "Metoprolol" akusonyeza okwanira efficacy mankhwalawa ndi sipekitiramu lonse la matenda a mtima, Pakati Tingaone m'mnyewa wamtima infarction, inatsekeratu mtsempha wamagazi matenda, arrhythmias a mitundu yosiyanasiyana, ndi othandiza ngati wothandizira prophylactic kuteteza zisadzachitikenso cha matenda a mtima.
Pharmacokinetic katundu "Betalok" malangizo mankhwala ntchito anafotokoza motere. Atalandira zayamba mankhwala onse mu nthawi yochepa ndipo odzipereka kwa mundawo m'mimba, ndende wake pazipita mu madzi ndi mfumukazi mwa ola limodzi kapena awiri. mankhwala akhoza mofulumira zimapukusidwa mu chiwindi, motero kutulutsa metabolites ndi pafupifupi palibe ntchito matupi chilichonse chamoyo. Hafu ya moyo mwa zigawo mankhwala ndi maola pafupifupi atatu kapena anayi, ndipo pafupifupi sasintha pa nthawi yonse ya mankhwala. Excretion wa metoprolol amapangidwa mu impso ndi - oposa 95% ya mlingo wa mankhwala, mmene zosaposa atatu peresenti excreted sichinasinthe.
"Betalok" mtsogoleri akuonetsa kuti nthawi ya matenda otsatirawa: zochizira matenda oopsa, monga nthumwi achire ntchito kuteteza zikwapu. mankhwala A tikuonera milandu arrhythmias mtima, komanso kupewa yachiwiri zofunika pambuyo akuvutika cardio-mtima dongosolo.
Mlingo kamwedwe wa Buku mankhwala "Betalok" malangizo akuonetsa kuti kukhazikitsa zimenezi. Mlingo pafupifupi mankhwala kawiri pa tsiku pa phwando mamiligalamu 100 pa tsiku. Nthawi zina, malangizo ikuti kuthekera kuwonjezeka pang'onopang'ono mlingo kawiri. Ngati mankhwala ntchito m'nsinga, mlingo umodzi zimasiyanasiyana 2 mpaka 5 mg. Ngati mu nkhani iyi si akwaniritsa anthu a mtima, lokonzekera angathe kuperekedwa mobwerezabwereza pambuyo Mphindi 5.
Mlingo kamwedwe ayenera kuganizira kuti ntchito mlingo pazipita mankhwala ndi 400 mg pa tsiku.
Pamene akulandira mankhwala "Betalok" Mwina kuyambitsa zotsatira zoyipa kwa kachitidwe zosiyanasiyana za thupi. Chotsatira awo mwatsatanetsatane ndi kufotokoza zizindikiro chikuperekedwa malangizo ntchito mankhwala.
Contraindications kulandira mankhwala osiyanasiyana malingana ndi mtundu ndi chikhalidwe cha otaya anatseka misewu mtima madutsidwe, hypotension, cardiogenic mantha ndi matenda ena. Contraindicated phwando ngati wodwalayo hypersensitivity kwa zigawo zake. Musawachite mankhwala pa mimba ndi yoyamwitsa.
Ndi kusamala kwambiri ayenera kulankhula kwa ntchito mankhwala ndi odwala COPD,
shuga, matenda Raynaud a.
Kuyima mankhwala osavomerezeka pang'onopang'ono, ndondomeko imeneyi ayenera masiku osachepera khumi.
Mankhwala angapo a modes wapadera wa kanthu, ndi kaphatikizidwe ndi mankhwala ena. Mfundozi zambiri amapezeka mu malangizo ntchito.
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