Thanzi, Kukonzekera
Haloperidol. Reviews kukonzekera bwino anayambitsa
Pakati pa nambala yaikulu ya mankhwala psychotropic neuroleptics zatenga malo kwambiri. Zikuphatikizapo "Haloperidol", ndemanga imene umboni nchito zake. Izi antipsychotic yogwira ntchito kwa zaka zambiri zochizira matenda ambiri amisala, kuphatikizapo akuchita misala. "Haloperidol" ali ndi zotsatira sedative ndi potentiates zotsatira za mankhwala, hypnotics ndi analgesics. The kanthu za mankhwala chifukwa cha kutchinga kwa noradrenergic Alpha chapakati ndi chachikulu kwambiri chapakati zolandilira dopamine. "Haloperidol" mtima umboni umene nthawi zina zoipa, nthawi zambiri kumayambitsa matenda extrapyramidal, amene Pamlingo waukulu chifukwa anatseka misewu ya maselo dopamine. Ndi zabwino antiemetic. Iye alibe zotumphukira ndi pakati anticholinergic kanthu.
"Haloperidol", ndemanga madokotala zomwe ndi zochokera nchito zake pothandiza onse a excitations thandizo lalikulu pamene wosangalala monyanyira limati ndi kuona zilubwelubwe. Ndi othandiza kuchiza odwala amene akhala akulimbana ndi atumiki antipsychotic. Mosiyana ndi mankhwala ena, sayambitsa ulesi ndi mphwayi, ndipo ali ndi mphamvu zotsatira. chida ichi Kwalamulidwa inati wosangalala monyanyira, schizophrenic psychoses, akhate limati onyenga pamene mwakwiya maganizo, involutional, oligophrenic, mowa psychoses epileptiform; matenda ena amagwirizana ndi kuyerekezera zinthu m'maganizo ndi psychomotor mukubwadamuka.
"Haloperidol", ndemanga pa ntchito zothandiza zimene mankhwalawa tremens kuona zilubwelubwe, limodzi ndi kuyerekezera zinthu m'maganizo zithunzi, ambiri mofulumira utatha motility ndipo kumatha masomphenya. Nthawi zambiri amatengedwa osakaniza analgesics, hypnotics ndi atumiki neurotropic kukonzekera wodwala kwa opaleshoni. Pali umboni akuthandiza mphamvu ya wothandizila pothandiza ululu, kunyansidwa ndi kusanza pa pachimake inatsekeratu insufficiency, wa malemeredwe. Ngati mankhwala antiemetic ntchito pa kusanza chiyambi iliyonse. Small Mlingo wa mankhwala ntchito limati zotakasika ndi neurotic.
"Haloperidol" zotchulidwa mkati (chakudya, makamaka mkaka) kapena jekeseni mu mnofu. Mlingo tsiku kumayambiriro kwa Inde - 1,5-3 mg. Odwala ndi kukana kuti wothandizila neuroleptic - 4-5 mg. mankhwalawa kuti analilembera Mlingo 3. Iwo Kwalamulidwa mapiritsi kapena madontho. Daily mlingo ndi chinawonjezeka ndi 0.5-2 mg, choncho kukaniza kwa 2-4 mg. Normal tsiku achire ranges mlingo wa 10-15 mg, ndi mitundu aakulu a akuchita misala kwa 20-40 mg. Muyezo nthawi Maphunzirowa - miyezi 2-3. kuchepetsa mlingo ayenera kukhala odekha. The tsiku yokonza mlingo - 0.5-5 mg. Ana osaposa zaka 5 ndi anatchulidwa kotala la mlingo wamkulu. Kuyambira zaka 6 mpaka 15 anaika theka la mlingo wamkulu. Gwiritsani ntchito sedative ndi, 0.5 mg, monga odana ndi - 1.5-2 mg.
Pali njira zina kupanga: mu phukusi la mapiritsi 50 (1.5 ndi 5 mg); 5 ampoules (1 ml) yankho la 0.5%; mu 10 ml Mbale (10 madontho = 1 mg).
Zovuta pambuyo ntchito: Parkinsonism, zotsatira dystonic, akathisia. Mpumulo wa mavuto Kwalamulidwa antiparkinsonian wothandizira.
Zotsatira zoyipa za mankhwalawa: galimoto mukubwadamuka, spasmodic chidule minofu thunthu, minofu nkhope; kumverera mantha ndi nkhawa; nseru; kusanza; otsika magazi; zochita khungu (toksikodermiya); kuchuluka tilinazo khungu ku dzuwa. "Haloperidol" amene ambiri osokoneza akhoza kuthetsa tulo yaitali, ayenera kumwedwa mosamala kwambiri ndi mankhwala ndi analgesics.
Contraindications: chipwirikiti, mantha ndi matenda a mtima. Haloperidol sayenera kugwiritsidwa ntchito pamene mowa.
Posachedwapa anaonekera mu mankhwala "Haloperidol decanoate" - yaitali wotenga mankhwala. Kukonza kupatula haloperidol kumaphatikizapo zitsamba mafuta ndi ethyl mowa.
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