Thanzi, Kukonzekera
"Clonazepam": ndemanga. "Clonazepam": malangizo ntchito, mavuto
"Clonazepam" - antiepileptic mankhwala limene limafotokoza kuti ena ofanana benzodiazepine. Pa polandira "clonazepam" mavoti otsalafe mankhwala makamaka positive. Mankhwala ali minofu anasiya ndipo zotsatira sedative, koma ali ndi zotsatira sedative.
The zikuchokera, amasulidwe mawonekedwe "clonazepam" mankhwala
Mankhwala alipo mapiritsi nkhani zosiyanasiyana zigawo zikuluzikulu:
- 0.5 mg. Kuwonjezera clonazepam, kapangidwe kumaphatikizapo lactose monohydrate. Kwa zosakaniza miyala likukhudza ndi sodium carboxymethylstarch. "Clonazepam" mapiritsi muli mankhwala enaake a stearate, gelatine. Auxiliaries alinso talc ndi wowuma mbatata. mapiritsi mtundu Ufumuyo utoto E110.
- 2 mg. Zina wothandiza zosakaniza - polysorbate 80, lactose monohydrate. The zikuchokera mankhwala pano carboxymethylstarch soda ndi sodium wochuluka lauryl sulphate. talc, gelatin ndi optional zosakaniza. Wothandiza zigawo zikuluzikulu ndipo ali ndi zinthu zina - mankhwala enaake a stearate, mpunga, mbatata wowuma.
Pharmacological kanthu "clonazepam" mankhwala
"Clonazepam" kumafooketsa pa ambiri nyumba amapanga dongosolo chapakati mantha, makamaka amene akukhudzana kugwira ntchito maganizo. Zotsatira za mankhwala "clonazepam" malangizo Buku, maganizo chimaonetsedwa monga sedative, anxiolytic ndi zachinyengo (lomaliza amtengo anafotokoza). The medicament kumachepetsa chigoba minofu kamvekedwe, kumathandiza zowombetsa mkota convulsive khunyu. Pali kulimbikitsa njira kuukira khunyu (focal, zowombetsa mkota).
Pharmacokinetics
mankhwala pafupifupi atamezedwa kotheratu ku kapepala m'mimba ndi outputted makamaka ndi impso (metabolites), gawo laling'ono (2%) limapezeka sichinasinthe. ndondomeko amatenga theka moyo wa maola 20 kuti 40. The bioavailability kukonzekera ingested ndi 90%, ubale ndi mwa kundipatsako magazi - 85%, ndende apamwamba anafika zikutanthauza maola 2.5. Mankhwalawa "clonazepam" zigawo zake kulowa mkaka wa m'mawere.
Zikuonetsa ntchito mankhwala
Miyala "clonazepam" oyenera zochizira odwala a zaka zosiyana ndi khunyu, kaya mawonetseredwe ake:
- khunyu tsankho (m'deralo, focal) wa digirii aliyense wa kusalekerera;
- zinthu convulsive (zimandilimbikitsa, clonic);
- khunyu yosavuta achiwiri zowombetsa mkota;
- amajomba atypical (Lennox-Gastaut syndrome);
- myoclonic kukomoka;
- lililonse pakalibe kukomoka;
- zimandilimbikitsa-clonic khunyu pulayimale ndi sekondale kuwonetseredwa.
"Clonazepam" zotchulidwa kuchepetsa minofu kamvekedwe, onse zachinyengo mavuto ndi psychomotor pa chithandizo.
Kugwiritsa ntchito mankhwala "clonazepam"
Mlingo chofunika anatsimikiza zochokera zifukwa zambiri. Pa siteji koyamba mankhwala amagwiritsa mlingo wochepa "clonazepam" (0.5 mg), pang'onopang'ono kusintha mlingo mpaka zotsatira anakhumba analandira. Pa nthawi yomweyo upambana mlingo pazipita ndikoletsedwa. Monga mauniko, "clonazepam" sangathe mwadzidzidzi kukwezedwa ngakhale pamene mankhwala anali sakhalitsa. Lakuthwa kukana mankhwala likuoneka chitukuko cha munthu kuyima khunyu.
Chikuonetseratu khunyu:
- Akulu. mankhwala koyamba imagwiridwa ntchito osapitirira 1 mg wa mankhwala. Mlingo masamu patsiku, ogaŵikana Mlingo 3 kapena 4, zimene ziyenera kuchitidwa fupipafupi. Popanda luso logwiritsa ntchito mankhwala pa mlingo wofanana, gawo lalikulu kwambiri "clonazepam" chakumwa asanagone. Childs, okwanira tsiku mlingo uli mu uthunthu wa 4 8 mg mankhwala. The yokonza mlingo sayenera upambana 20 mg (akwaniritsa pa masabata 2-4 mankhwala). Pamene anatsimikiza tsiku mlingo ogwira, amene amalola kukhala chikhalidwe zachibadwa za thupi, izo amaloledwa mlingo umodzi pogona.
- Ana (ndi kulemera kwa osachepera 30 kg). Monga mauniko, "clonazepam" poyambirira anasonyeza ana 0.5 mg ndi kudziwa mlingo wake mulingo woyenera.
Phwando ndi matendawa, amene anatsagana ndi ululu paroxysmal:
- Akulu. Choyamba, odwala kutumikiridwa 1-2 tsiku dosing (0.5 mg wa nthawi iliyonse). odwala ambiri okwanira achire mlingo ndi 1 mg / tsiku. Tsiku sangathe kumwa kuposa 1 mg wa mankhwala "clonazepam". Reviews Komabe, kusonyeza kuti nthawi zina, madokotala achuluke mlingo 4 mg. Zikatero, mlingo ali anasintha pang'onopang'ono (osiyanasiyana - masiku 3, mwina kuwonjezera 0.5 mg). Pamene mukufuna kuchepetsa zovuta tulo masana, mlingo masamu pa phwando masana, inu kukhoza pamaso yogona.
- Ana. Kwa odwala amene sali zaka zoposa 18, kudziwika vuto mankhwala akhoza kukhala operewera ndi woopsa.
Kupewa mavuto alionse, mankhwala "clonazepam" ndemanga Madokotala amalangiza kutenga mosamalitsa pa malangizo a katswiri amene achitila.
Contraindications kulandira "clonazepam" mankhwala
Mapiritsi sizigwiritsidwa ntchito pamene kuchuluka kudziwa zinthu imene iwo analemba. mankhwala ali contraindicated mu maiko awa:
- myasthenia gravis;
- kuwonongeka kwa chikumbumtima;
- wobereka, kuyamwitsa;
- khungu (kutsekedwa);
- matenda kupuma kukhala chiyambi chapakati, aakulu kupuma insufficiency;
- Lolemera umayenda aimpso ndi kwa chiwindi kulephera;
- kuwonekera kwa matenda matenda obanika kutulo;
- mowa poizoni;
- porphyria pachimake mawonekedwe.
Zotsatira zoyipa "clonazepam" mankhwala
Taganizirani mavuto, yomwe INGATHE kuyambitsa "clonazepam". Ntchito mankhwala akhoza kugwirizana ndi zochita chowawa. Zikhoza ulesi, nseru, irritability. Ngati anakwiya ndi thupi amatopa msanga, iye wakhala kugwirizana kayendedwe. Kuchepetsa zotsatira za kuonekera mavuto, choyamba muyenera kutsatira mlingo yaing'ono, pang'onopang'ono kuwonjezeka kufikira izo zitakhala mulingo woyenera.
Amadziwika kuti pa chithandizo "clonazepam" amatanthauza ntchito ndi kuphwanya malangizo zingachititse ambiri osokoneza. Zikatero, pali zidzasintha, tingayambe chisokonezo, stupor, zomwe zingadzetse chikomokere. Mwa zizindikiro zina - mtima kugwa, mkhutu kupuma, kusinza. M'pofunika kusambitsana m'mimba (mwaluso yomweyo pambuyo wonyeketsa mapiritsi) kuchititsa mankhwala oyenera. Nkofunika nthawi zonse kuyan'ana kusintha zizindikiro monga magazi, zimachitika, kupuma. Nthawi zina, pamafunika kukhazikitsa mpweya makina. Pali mankhwala - "Flyumazenil," koma si oyenera makonzedwe odwala amene akukuchitirani "clonazepam" kwa nthawi yaitali.
Sikuti kuphatikiza "clonazepam" ndi mowa. Reviews kulola onetsetsani kuti kuphatikiza akhoza kusokoneza moyo. N'chimodzimodzinso ndi mankhwala zonse kuchita chapakati mantha dongosolo, inhibiting ntchito yake.
mogwirizana mankhwala "clonazepam" kukonzekera
Zotsatira za mankhwala kuwonjezera analgesics chomwa mankhwalawa, anticonvulsants. The chifukwa chomwecho zimawonedwa ndi kaphatikizidwe ndi antidepressants, neuroleptics, barbiturates, komanso pamene pamodzi ndi mowa ndi zinthu musawachitire chigoba minofu kamvekedwe. Mphamvu ya mankhwala yafupika pamene ingested chikonga.
Cost, ndemanga za mankhwala "clonazepam"
Gulani "clonazepam" mapilitsi mu Moscow kungakhale kwa 97-150 rubles. (30 ma PC.). Mankhwala othandiza mu khunyu, ngati anamvera kuimilidwa ndi dokotala. Pamene atonic kukomoka mwina miyezi iwiri, nthawi ya mankhwala chikukwanira nthawi yotero, mukhoza kusinthana kwa chithandizo yokonza. Nthawi zina pali mavuto, koma makamaka okha koyamba gawo wa mankhwala, nthawi zambiri kufooka.
Tikayang'ana mudziwe kuti muli ndi ndemanga, "clonazepam" kamakhala kuchotsa chinawonjezeka minofu kamvekedwe mu pafupi masabata atatu. Madokotala mwina mankhwala ngati alamu, mantha, IRR, amene anatsagana ndi amantha. Mankhwala othandiza, ntchito msanga.
Reviews "clonazepam" chimaonetsedwa monga njira zabwino kuti amachita ntchito yake, koma zingachititse kuti amadwaladwala (kufooka, kutopa, ndi zina zotero. P.).
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