Thanzi, Kukonzekera
"Siofor 500"
"Siofor 500" - mankhwala omwe amagwiritsidwa ntchito kuchepetsa miyeso ya magazi m'magazi kwa odwala matenda a shuga. Mankhwalawa amapangidwa pokhapokha mu mawonekedwe a piritsi, amaphimbidwa ndi chovala chapadera ndipo amalinganiza kuti alowemo mkati.
Mankhwala omwe amagwiritsidwa ntchito pokonza "Siofor 500" ndi metformin hydrochloride. Zothandizira zothandizira zikuphatikizapo magnesium stearate, povidone, hypromellose, titaniyamu ya dioxide, macrogol 6000.
Kuchita zachipatala kwa mankhwala awa ndi chifukwa chokhala m'gulu la a biguanide. Mukalowetsa magazi mwachindunji, amawonetsa mphamvu ya hypoglycemic (kuchepetsedwa kwa ndondomeko ya shuga). "Siofor 500" sichikhudza kugwira ntchito kwapasitiki, choncho zikachitika, mlingo wa insulini sukusintha. Mankhwala ofanana ndi metformin amaletsa glycogenolysis ndi gluconeogenesis, kotero kupangidwa kwa shuga mu maselo a chiwindi kuchepetsedwa. Zimathandizanso kuti minofu ikhale yotetezeka ku insulini, imalepheretsa kuyamwa kwa mankhwalawa m'matumbo. Zotsatira zofanana nthawi zina zimalola kugwiritsa ntchito "Siofor 500" polemera. Mankhwalawa ali ndi zinthu zina zothandiza, zomwe zimaphatikizapo kukakamizidwa kwa mavitamini a glycogen, kuwonjezeka kwa kayendedwe ka mapuloteni a shuga, kumachepetsa mlingo wa kolesterolini, triglycerides.
Mankhwala osokoneza bongo atatha kumwa amawoneka pambuyo pa maola awiri. Kudya chakudya kumachepetsa chizindikiro ichi. Mndandanda wa bioavailability ndiwo makumi asanu peresenti. Mankhwalawa amatulutsidwa mu mkodzo. Half-moyo wa zigawo zonse ndi ola limodzi ndi theka. Pomwe kuchepa kwa impso kumachepa, chizindikiro ichi chikuwonjezeka. Kuonjezera apo, mankhwala a plasma a mankhwala othandiza amawonjezera mankhwala.
Mlingo wa mankhwala umatsimikiziridwa payekha. Zimatsimikiziridwa ndi msinkhu wamagulu a m'magazi. Chithandizo chikuchitika malinga ndi mfundo ya kukula kwa mlingo. Mankhwalawa ayenera kutengedwa pakudya, kutsukidwa ndi madzi ochulukirapo, osasaka. Ulamuliro wa nthawi ziwiri ndi wotheka pa mlingo womwe uli piritsi limodzi patsiku. Kutalika kwa mankhwalawo kumatsimikiziridwa ndi dokotala. Kudya mankhwala osokonezeka sikungathe kulipiritsika pogwiritsira ntchito mapiritsi ambiri. Mlingo wa mankhwalawo uyenera kuchepetsedwa nthawi yomweyo pamene matenda amadzimadzi amapezeka.
"Siofor 500" ndi mankhwala omwe ayenera kugwiritsidwa ntchito poyang'anira dokotala. Nthawi zina mavuto amayamba, kuphatikizapo lactacidosis, matenda opuma, kufooka, kusanza, kunyowa, kugona, kutsekula m'mimba, hypothermia, kupweteka kwa m'mimba, kuchepa kwa mtima, kusokonezeka, kutaya mtima. Kuonjezera apo, zochitika zomwe zimachitika m'magazi a megaloblastic, kusokonezeka maganizo.
Pomwe dokotala akufunsana, m'pofunika kufotokoza zotsutsana ndi kugwiritsa ntchito mankhwala. Ambiri ali ndi shuga ya ketoacidosis, omwe amachititsa kuti munthu asagwiritsidwe ntchito molakwika, asagwiritsidwe ntchito mopitirira muyeso, amatha kusokonezeka m'mtima, matenda osokoneza bongo, matenda, matenda opatsirana, opaleshoni, kapangidwe ka munthu. Ndiletsedwa kugwiritsa ntchito mankhwalawa masiku angapo musanayambe maphunziro a radioisotope.
Chotsutsana kwambiri ndi kugwiritsa ntchito mankhwalawa ndi nthawi ya mimba, lactation. "Siofor" ndi mowa sagwirizana, kuphatikiza kumeneku kungayambitse chitukuko chachikulu cha matenda opatsirana, chomwe chichotsedwe chomwe chidzafuna kuthetseratu zinthu zowononga ndi kugwiritsa ntchito mankhwala opatsirana.
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